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| Year | Name | Affililiation |
| 1957 | Prof. J.M. Bijvoet | University of Utrecht, the Netherlands |
| 1962 | Prof. A.R. Ubbelohde | Imperial College of Science and Technology London, UK |
| 1968 | Prof. V. Prelog | Technische Hochschule Zürich, Switzerland |
| 1974 | Prof. L.J. Oosterhoff | University of Leiden, the Netherlands |
| Prof. W.S Johnson | Stanford University, USA | |
| Prof. J.M. Lehn | University of Strasbourg, France | |
| Prof. W.N. Lipscomb | Harvard University, USA | |
| 1978 | Prof. E. Havinga | University of Leiden, the Netherlands |
| 1983 | Prof. M. Karplus | Harvard University, USA |
| 1988 | Prof. J.M. Thomas | Royal Institute of Great Britain London, UK |
| 1994 | Prof. R. Breslow | Columbia University New York, USA |
| 1998 | Prof. E.N. Jacobsen | Harvard University, USA |
| 2001 | Prof. M.T. Reetz | Max Planck Institut Mühlheim, Germany |
|
Prof. J.M. Lehn |
Prof. E.W. Meijer Collège de France Paris, France | |
| Prof. P.W. Atkins | Oxford University, UK | |
| Prof. E.W. Meijer | Eindhoven University of Technology, the Netherlands | |
| 2004 | Prof. G.M. Whitesides | Harvard University, USA |
| 2009 |
Prof. D.W.C. MacMillan |
Princeton University, USA |
| Prof. T. Carell | Ludwigs-Maximillians-University Munich, Germany | |
| Prof. J. Aizenberg | Harvard University, USA | |
| Prof. B.L. Feringa | University of Groningen, the Netherlands | |
| 2011 | Prof. S.L. Schreiber | Harvard University, USA |
| Prof. C.A. Mirkin | Northwestern University, USA | |
| Prof. C. Robinson | Oxford University, UK |
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